HM15211 LAPS
PT-141, measured in a single radioligand displacement series against I-NDP-alpha-MSH on membranes from BHK570 cells stably expressing each human subtype, returned Ki 0.25 nM at MC4R, 6.4 nM at MC1R, 17 nM at MC5R and 53 nM at MC3R, roughly 26-fold, 68-fold and 210-fold preference for MC4R over MC1R, MC5R and MC3R respectively
Derrien, M., Belzer, C
For instance, this peptide is very much loved by those who are fond of tanning but do not want to expose themselves to the sun or a tanning bed for a long time, hence minimizing the risk of getting charred
Initial pricing sets the 1.5mg and 4mg doses at $149 per month, with changes planned after April 15, 2026: the 4mg dose rising to $199 and higher maintenance doses (9mg and 25mg) priced at $299 per month
District Court for the Southern District of Florida